Lesi sidakamizwa sinempahla ye-vasodilator, i-anticonvulsant kanye ne-antihypertensive. Isenzo saso esisheshayo kufanele sigcwalise ukumuncwa emzimbeni. Amaphilisi e-Papaverine anciphisa ithoni yezinsipho ezibushelelezi, ukwandisa imishanguzo, ukwandisa ukugeleza kwegazi, ngaleyo ndlela ukunciphisa ubuhlungu be-spastic.
Ukwakhiwa kwamaphilisi e-papaverine
Ingxenye eyinhloko yamaphilisi i-papaverine hydrochloride (10 mg nge-tablet ngayinye). Izinto ezisizayo zifaka isitashi sezambane, i-stearic acid, ishukela elicwengekile ne-talc.
Izinkomba zokusebenzisa amaphilisi e-papaverine
Isenzo sesidakamizwa singenxa yokuvinjelwa komsebenzi we-phosphodiesterase enzymes etholakala emisipha. Ngenxa yalokhu, akunakwenzeka ukwakha i-actomiosin kuzicubu zeprotheni, okuyinto engxenyeni eyinhloko ephethe ukuhlukunyezwa kwemisipha.
Umuthi unqunywe kula macala alandelayo:
- ukuqeda izicathulo zemisipha ebushelelezi, okuholela ekusenikeni kobuhlungu besifo;
- ekucindezelekeni okuphakanyisiwe ukuthi yisiphi isizathu se-articulation of arteries kanye nokumelana okukhulu kodonga lwezitsha;
- kwi-anesthesiology yokulungiselela;
- abesifazane abakhulelwe ngezwi elikhudlwana lesibeletho .
Ukungahambisani nokusetshenziswa kwamaphilisi e-papaverine
Ukwelashwa ngalesi sidakamizwa kuvunyelwe amaqembu alandelayo abantu:
- izingane kuze kube izinyanga eziyisithupha;
- abantu asebekhulile;
- ukuhlukunyezwa kwesibindi;
- ube ne-glaucoma;
- izingxenye ezingahambisani nomuthi.
Ngokuqapha kufanele kuthathwe ezimweni ezinjalo:
- i-hypothyroidism;
- ngemuva kokulimala kokuchofoza ebuchosheni;
- ne-tachycardia engaphezulu;
- esimweni sokushaqeka;
- ngokuhluleka kwezintambo zesimo esingapheliyo;
- nge-prostatic hyperlasia.
Abesifazane abakhulelwe kufanele babonane nodokotela.
Ungathatha kanjani i-papaverine kumaphilisi?
Isidakamizwa sitholakala kumathebulethi angu-40 mg. Kukhona futhi uhlobo lokukhululwa kwabantwana abangu-10 mg. Thatha izikhathi ezintathu ngosuku (kungakhathaliseki isikhathi sokudla). Uma isingenwe, isidakamizwa sisatshalaliswa ngokweqile kuma-tissue. I-excreted kanye nomchamo ngendlela yemikhiqizo ye-metabolism yesibindi.
Njengoba lesi sidakamizwa sincipha kancane kancane emzimbeni, umphumela wayo awuhambisani nezezinye ze-antispasmodics, njenge- No-shpa . Ukubhekana nobuhlungu obukhulu uPataverin uyasiza kuphela, ngakho-ke ukuthuthukisa umphumela okunconywa ukuthatha neminye imithi yobuhlungu - i-Aspirin noma iParacetamol.