Spray Izoket (eJalimane) ibhekisela ezidakamizweni ze-vasodilator ezivela eqenjini le-nitrate ephilayo. Isidakamizwa sinciphisa umthwalo esikhungweni se-myocardium, ukunciphisa isidingo senhliziyo yomzimba ngamandla ne-oxygen. Isixazululo esingenambala se-Isoket sigcwele amabhodlela angenalutho engilazi engama-15 ml, enesisipuni se-dispenser-sprayer. Uma usebenzisa i-aerosol, i-pump mechanical iqala. Kubalulekile ukuthi i-freon, eyingozi emkhathini, ayisetshenziswanga ku-aerosol.
Ukwakhiwa kwe-Isoket yomkhiqizo
Into esebenzayo eyinhloko, equkethwe kumithi yokwelapha, i-isosorbide dinitrate inezakhiwo ze-vasodilating. Ngaphezu kwalokho, ukwakheka kwefomu le-aerosol yomuthi Izoket kuhlanganisa i-ethanol ne-macrogol-400.
Isicelo se-Isoket Spray
Njengendlela yokwelapha i-Isoket ekhethiwe:
- ngenhloso yokuboshwa kwe-angina pectoris ;
- ukuvimbela ukuhlaselwa kwe-stenocardia;
- ne-infarction ye-myocardial;
- esikhathini esilandelayo.
Imithetho yohlelo lokusebenza lwe-Isoket Spray
I-Aerosol isoket isetshenziswa ngendlela elandelayo:
- Ibhodlela elinomuthi litholakala ngokuqondile.
- Idivaysi yokulinganisa itholakala eduze nesigxobo somlomo.
- Ukuphefumula okujulile kuthathwa, kulandelwa ukubambezeleka kokuphefumula.
- Ukucindezelwa kwesikhathi esisodwa ku-nebulizer kwenziwa, futhi into engena emlonyeni womlomo.
- Kudingeka ukuvala umlomo wakho kanye nemizuzwana engu-30 ukuphefumula ngekhala lakho.
Ukunakwa sicela! Ngama-angina afanelekayo noma okusolakala ukuthi i-infarction enomsoco, udokotela angase akhulise umthamo ophakanyisiwe wesidakamizwa izikhathi ezingu-2 kuya kwezi-3. Uma isiguli singathuthuki, inqubo ingabuyekezwa emva kwemizuzu emihlanu.
Gwema ukuthola Isoket emehlweni!
Ukuqhathaniswa nokusetshenziswa kwe-Isoket ye-spray
Isidakamizwa sinokuphikisana okuningi, ngakho-ke, i-Isoket ivunyelwe ukusebenzisa uma:
- ukungakwazi kahle kwamathambo;
- I-hypotension ye-arterial (uma ingcindezi ingaphansi kuka 90/60);
- i-glaucoma ehlukahlukene-evaliwe;
- ukuphazamiseka kwengqondo;
- i-hyperthyroidism;
- ukuntuleka kwe-glucose-6-phosphate dehydrogenase;
- ukuzwela ngokweqile ezingxenyeni zomuthi, ngokuyinhloko ukuba isosorbide nitrate.
Ngokuqapha, i-aerosol kufanele isetshenziselwe ukuphazamiseka kokusebenza kwezinso nesibindi. Kuyinto engathandeki ukusebenzisa i-Isoket ekwelapheni kwezingane kanye nentsha engaphansi kweminyaka engu-18 ngenxa yolwazi olunganele mayelana nokuphepha kwesidakamizwa semvelo ekhulayo. Ungasebenzisi i-Isoket Spray kanyekanye ne-phosphodiesterase hlobo 5 inhibitors (uSildenafil nokunye). Ngesikhathi sokukhulelwa ne-lactation, lesi sidakamizwa singabekwa kuphela ezimweni lapho inzuzo engaba khona kowesifazane kusukela ekusebenziseni kwayo kudlula ingozi yempilo yengane noma ingane.
Kukhona ubufakazi bokuthi ukuthatha i-Izote kungaholela ekuphazamiseni ikhono lokushayela izimoto.
Sula i-Isoket ye-analogues
Esinye sezifanekiselo ezithandwayo ze-Isoket yezidakamizwa nayo imishanguzo yaseJalimane iKardiket. Shintsha i-Isoket e-spray ingaba yisisombululo se-Isoket, amafomu e-aerosol okukhipha ukumnika i-Nitrosprey (eRussia),
- I-Nitrosorbide;
- I-Nitrosorbid NS;
- I-nitrosobid-Rusfar;
- I-Nitrosorbide-UVI.
Izindleko zemishini yokukhiqiza yaseRashiya naseHungary ziyi-3-4 izikhathi eziphansi, kanti amaphilisi e-NitroSorbide aphansi kakhulu kunalokho okufakwe kwe-Isoket okufakiwe.
Ngesikhathi esifanayo, izazi zithi amafomu e-aerosol anomphumela osheshayo futhi anikeze isikhathi esiphezulu sethonya kunamaphilisi namaphissile anomphumela ofanayo.